Pending final data from our Phase 1 trial of APG777 in healthy volunteers, we may initiate a Phase 2 trial in asthma and expect to further evaluate opportunities to develop APG777 for other I&I indications, including alopecia areata, chronic rhinosinusitis with nasal polyps, chronic spontaneous urticaria, eosinophilic esophagitis and prurigo nodularis.
(1)Our philosophy is simple.
Our goal is to discover and develop new differentiated therapies for a range of I&I indications. We aim to accomplish this goal by focusing on known biologic drivers of disease and utilizing advanced antibody engineering to develop product candidates with optimized properties that have the potential to overcome limitations of existing therapies. We believe our approach will enable us to develop a portfolio of therapies that are differentiated compared to the currently available standards of care and address unmet medical needs for I&I indications.
Pipeline
STRATEGY
PROGRAM
Discovery
PRE-CLINICAL
PHASE 1
PHASE 2
PHASE 3
NEXT ANTICIPATED MILESTONES
Best-in-class monotherapy in AD
Higher exposures for better efficacy with less frequent dosingIL-13
APG777- 2H 2025: Phase 2 16-week induction PoC data
Best-in-class mAbs for combinations
Strategic optionality to combine orthogonal mechanisms across pipelineIL-4Rα
APG808- Q4 2024: Initial Phase 1 PK and safety in HVs
OX40L
APG990- 1H 2025: Initial Phase 1 PK & safety in HVs
TSLP
APG333- Late 2024 / Early 2025: Initiate Phase 1 PK & safety in HVs
First- or best-in-class combination approaches
Rational combinations to drive broader + deeper responsesIL-13 ± OX40L
APG777 ± APG990- 2025: Clinical trial initiation
IL-13 ± TSLP
APG777 ± APG333- TBD: Clinical trial initiation1
IL-13/IL-4RΑ + OX40L/TSLP
ADDITIONAL COMBINATION(S)- December 2, 2024: Additional combination(s) to be announced at R&D Day